Skip to main content

binimetinib

Generic: BINIMETINIB·Brand: MEKTOVI, Mektovi

binimetinib: developed by 1 company · 16 clinical trials tracked · 1 FDA decision.

binimetinib evidence translation

What we can confirm

1 FDA record · 16 tracked trials

What it means

Source-backed records connect binimetinib to ARRY; that link alone does not prove the drug works.

What to watch

Watch active trials and any change in FDA or trial status.
BioSniper AIPage evidence connected

Prepared research question

How could binimetinib → ARRY affect its developer, and what evidence supports the link?

Run cited research

Traceable citations · Unknowns marked

See linked entities and source evidence8 indications · 7 study sponsors
Development Pipeline (1)
CompanyPhase
ARRAY BIOPHARMA INC (ARRY)
unresectable or metastatic melanoma with a BRAF V600E or BRA…
Approved
Clinical Trials (16)showing 10 most recent

Molecular Targeted Maintenance Therapy Versus Standard of Care in Advanced Biliary Cancer: an International, Randomised, Controlled, Open-label, Platform Phase 3 Trial

NCT05615818·Phase 3
Recruiting

Primary endpoint: Progression-free survival (PFS)

InterventionalRandomizedopen800 targetStarted 2024-07Completion 2028-0650 sites · Belgium, France, United KingdomUNICANCER

FOLFOX in Combination With Binimetinib as 2nd Line Therapy for Patients With Advanced Biliary Tract Cancers With MAPK Pathway Alterations: A ComboMATCH Treatment Trial

NCT05564403·Phase 2·BBOT
Active, not recruiting

Primary endpoint: Overall survival (OS)

InterventionalRandomizedopen66 targetStarted 2024-02Completion 2026-0550 sites · United StatesNational Cancer Institute (NCI)

Molecular Analysis for Combination Therapy Choice (ComboMATCH)

NCT05564377·Phase 2·RLAY
Recruiting

Primary endpoint: Accrual of patients to ComboMATCH treatment trials

InterventionalRandomizedopen2,900 targetStarted 2023-04Completion 2030-0750 sites · United StatesNational Cancer Institute (NCI)

A Phase 1 Study of ZEN003694 in Combination With Binimetinib in Solid Tumors With RAS Pathway Alterations and Triple Negative Breast Cancer

NCT05111561·Phase 1·RLAY
Suspended

Primary endpoint: Incidence of dose limiting toxicities (Part 1 [Dose Escalation])

Interventionalopen42 targetStarted 2022-08Completion 2027-034 sites · United StatesNational Cancer Institute (NCI)

A PHASE 1, OPEN-LABEL, DOSE ESCALATION AND DOSE EXPANSION STUDY TO EVALUATE THE SAFETY, TOLERABILITY, PHARMACOKINETICS, AND ANTI TUMOR ACTIVITY OF PF-07799933 (ARRY-440) AS A SINGLE AGENT AND IN COMBINATION THERAPY IN PARTICIPANTS 16 YEARS AND OLDER WITH ADVANCED SOLID TUMORS WITH BRAF ALTERATIONS

NCT05355701·Phase 1·PFE
Recruiting

Primary endpoint: Number of participants with dose limiting toxicities (DLTs) (Part 1 and Part 2)

Interventionalopen267 targetStarted 2022-07Completion 2029-1040 sites · Canada, Israel, United StatesPfizer

A Phase 1 Study of Nilotinib in Combination With Dabrafenib and Trametinib or Encorafenib/Binimetinib in BRAF V600 Mutant Metastatic Melanoma After Progression on BRAF/MEK Inhibition

NCT04903119·Phase 1·NVS
Recruiting

Primary endpoint: Percentage of Patients Experiencing Dose Limiting Toxicities

Interventionalopen30 targetStarted 2022-06Completion 2030-064 sites · United StatesRina Plattner

A Phase II Study of Binimetinib Plus Belinostat for Subjects With Metastatic Uveal Melanoma

NCT05170334·Phase 2
Active, not recruiting

Primary endpoint: Overall Response Rate

Interventionalopen7 targetStarted 2021-12Completion 2028-011 site · United StatesH. Lee Moffitt Cancer Center and Research Institute

A Phase II Neoadjuvant Study of Encorafenib With Binimetinib in Patients With Resectable Locoregional Metastases From Cutaneous or Unknown Primary Melanoma (Stages III N1B/C/D)

NCT04221438·Phase 2
Terminated

Primary endpoint: Pathologic Complete Response

Interventionalopen3 enrolledStarted 2021-09Completion 2025-0110 sites · United StatesECOG-ACRIN Cancer Research Group

A Phase 1/2, First-in-Human Study of DCC-3116 as Monotherapy and in Combination With RAS/MAPK Pathway Inhibitors in Patients With Advanced or Metastatic Solid Tumors With RAS/MAPK Pathway Mutations

NCT04892017·Phase 1·DCPH
Terminated

Primary endpoint: Incidence of Adverse Events

Interventionalopen91 targetStarted 2021-06Completion 2026-0310 sites · United StatesDeciphera Pharmaceuticals, LLC

A Phase II Study of Binimetinib in Combination With Imatinib in Patients With Advanced KIT-Mutant Melanoma

NCT04598009·Phase 2
Recruiting

Primary endpoint: Objective response rate (ORR)

Interventionalopen25 targetStarted 2021-03Completion 2028-052 sites · United StatesUniversity of California, San Francisco
FDA Decisions1 records
Approval1 INDICATIONS AND USAGE MEKTOVI is a kinase inhibitor indicated: • in combination with encorafenib, for the treatment of patients with unresectable or metastatic melanoma with a BRAF V600E or V600K mutation, as detected by an FDA-approved test. ( 1.1 , 2.1 ) • in combination with encorafenib, for the treatment of adult patients with metastatic non-small cell lung cancer (NSCLC) with a BRAF V600E mutation, as detected by an FDA-approved test. ( 1.2 , 2.1 ) 1.1 BRAF V600E or V600K Mutation-Positiv(ARRY)FDA ↗
NDA210498Type 1 - New Molecular EntityOrphan DrugStandardOralTablet

Frequently asked questions

Who is developing binimetinib?

binimetinib is being developed by ARRAY BIOPHARMA INC.

How many clinical trials involve binimetinib?

BioSniper tracks 16 clinical trials involving binimetinib.

What is binimetinib's latest FDA decision?

The most recent tracked FDA decision for binimetinib is Approval for 1 INDICATIONS AND USAGE MEKTOVI is a kinase inhibitor indicated: • in combination with encorafenib, for the treatment of patients with unresectable or metastatic melanoma with a BRAF V600E or V600K mutation, as detected by an FDA-approved test. ( 1.1 , 2.1 ) • in combination with encorafenib, for the treatment of adult patients with metastatic non-small cell lung cancer (NSCLC) with a BRAF V600E mutation, as detected by an FDA-approved test. ( 1.2 , 2.1 ) 1.1 BRAF V600E or V600K Mutation-Positiv, dated June 27, 2018.