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sapanisertib

Generic: sapanisertib

sapanisertib: developed by 1 company · 4 clinical trials tracked.

sapanisertib evidence translation

What we can confirm

What it means

Source-backed records connect sapanisertib to CALA; that link alone does not prove the drug works.

What to watch

Watch trial status, endpoints, and the next source-backed update.
BioSniper AIPage evidence connected

Prepared research question

How could sapanisertib → CALA affect its developer, and what evidence supports the link?

Run cited research

Traceable citations · Unknowns marked

See linked entities and source evidence8 indications · 2 study sponsors

Related indications

Squamous non-small cell lung cancer (sqNSCLC) harboring NRF2 (NFE2L2) mutations; evaluation also in NRF2 wild-type sqNSCLC and potential exploration in KEAP1-mutant tumors and KEAP1/NRF2 mutant tumor types beyond NSCLCOncology - being evaluated in NRF2-mutated sqNSCLCBreast CarcinomaCervical CarcinomaColorectal CarcinomaEndometrial CancerEndometrial CarcinomaGlioma
Development Pipeline (2)
CompanyPhase
Calithera Biosciences, Inc. (CALA)
Squamous non-small cell lung cancer (sqNSCLC) harboring NRF2…
Phase 2
Calithera Biosciences, Inc. (CALA)
Oncology - being evaluated in NRF2-mutated sqNSCLC
Phase 2
Clinical Trials (4)

Open-Label Umbrella Study to Evaluate Safety and Efficacy of Sapanisertib and Serabelisib (PIKTOR) in Various Combinations in Patients With HR+/HER2- Advanced or Metastatic Breast Cancer

NCT07558733·Phase 1/Phase 2
Recruiting

Primary endpoint: Safety and tolerability of drugs by assessment of adverse events (AEs) / serious adverse events (SAEs)

Interventionalopen32 targetStarted 2026-04Completion 2033-057 sites · United StatesFaeth Therapeutics

A Phase I/II Trial of Sapanisertib in Combination With Cabozantinib in β-catenin-mutated Hepatocellular Carcinoma (SAPHIRE)

NCT06811116·Phase 1·RPRX
Recruiting

Primary endpoint: Dose-limiting toxicities and incidence of adverse events

InterventionalRandomizedopen92 targetStarted 2025-11Completion 2027-084 sites · United StatesNational Cancer Institute (NCI)

An Open-label, Multi-Center, Phase 2 Clinical Trial Evaluating Sapanisertib and Serabelisib (PIKTOR) With Paclitaxel, and a Substudy Evaluating PIKTOR With Paclitaxel Plus an Insulin-Suppressing Diet, in Patients With Advanced or Recurrent Endometrial Cancer

NCT06463028·Phase 2
Recruiting

Primary endpoint: Objective Response Rate (ORR)

Interventionalopen40 targetStarted 2024-12Completion 2029-0918 sites · United StatesFaeth Therapeutics

Molecular Analysis for Therapy Choice (MATCH)

NCT02465060·Phase 2·ADMA
Active, not recruiting

Primary endpoint: Objective response rate (ORR)

Interventionalopen6,452 targetStarted 2015-08Completion 2026-1250 sites · United StatesNational Cancer Institute (NCI)

Frequently asked questions

Who is developing sapanisertib?

sapanisertib is being developed by Calithera Biosciences, Inc..

How many clinical trials involve sapanisertib?

BioSniper tracks 4 clinical trials involving sapanisertib.