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pan-mutant-selective pi3k-alpha inhibitor rly-5836

Generic: Pan-mutant-selective PI3K-alpha Inhibitor RLY-5836

pan-mutant-selective pi3k-alpha inhibitor rly-5836: 1 clinical trial tracked.

pan-mutant-selective pi3k-alpha inhibitor rly-5836 evidence translation

What we can confirm

1 tracked trial

No verified listed company relationship

What it means

AI will separate confirmed drug evidence from unknown company context.

What to watch

Watch trial status, endpoints, and the next source-backed update.
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Prepared research question

What is verified about pan-mutant-selective pi3k-alpha inhibitor rly-5836, and what remains unknown?

Run cited research

Traceable citations · Unknowns marked

See linked entities and source evidence3 indications · 1 study sponsors
Clinical Trial Registry Records (1)

A First-in-Human Study of PI3Kα Inhibitor, RLY-5836, in Combination With Targeted and Endocrine Therapies in Participants With Advanced Breast Cancer and as a Single Agent in Advanced Solid Tumors

NCT05759949Registry updated 2025-05-16·Phase 1·RLAY
Completed

Primary endpoint: Maximum Tolerated Dose (MTD) and Recommended Phase 2 Dose (RP2D) of RLY-5836

Interventionalopen41 enrolledStarted 2023-03Completion 2025-047 sites · United StatesRelay Therapeutics, Inc.