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azenosertib

Generic: ZN-c3·Code: ZN-c3

azenosertib: developed by 1 company · 9 clinical trials tracked.

azenosertib evidence translation

What we can confirm

What it means

Source-backed records connect azenosertib to ZNTL; that link alone does not prove the drug works.

What to watch

Watch trial status, endpoints, and the next source-backed update.
BioSniper AIPage evidence connected

Prepared research question

How could azenosertib → ZNTL affect its developer, and what evidence supports the link?

Run cited research

Traceable citations · Unknowns marked

See linked entities and source evidence8 indications · 0 study sponsors

Study sponsors

No additional listed-company sponsor is linked.

Development Pipeline (1)
CompanyPhase
Zentalis Pharmaceuticals, Inc. (ZNTL)
Solid Tumor; Osteosarcoma; Uterine Serous Carcinoma
Phase 3
Clinical Trials (9)

A Randomized, Open-Label Phase 3 Study of Azenosertib Versus Investigator's Choice of Chemotherapy in Platinum-Resistant High-Grade Serous Ovarian, Primary Peritoneal, or Fallopian Tube Cancers Positive for Cyclin E1 Protein Expression

NCT07546500·Phase 3·ZNTL
Recruiting

Primary endpoint: Progression free survival (PFS) per RECIST v1.1 as assessed by Investigator

InterventionalRandomizedopen420 targetStarted 2026-04Completion 2030-0450 sites · Australia, Belgium, Canada, France…K-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

A Phase I/II Single-arm Trial of Azenosertib (ZN-c3) Combined With Carboplatin and Pembrolizumab in Patients With Metastatic Triple-negative Breast Cancer (ZAP-IT)

NCT06351332·Phase 1
Terminated

Primary endpoint: Number of Participants Experiencing Dose Limiting Toxicity (DLT)

Interventionalopen7 targetStarted 2024-05Completion 2026-021 site · United StatesFilipa Lynce, MD

A Phase 2 Open-Label, Multicenter Study To Evaluate Efficacy And Safety Of ZN-c3 In Subjects With High-Grade Serous Ovarian, Fallopian Tube, Or Primary Peritoneal Cancer (DENALI / ZN-c3-005 / GOG-3066)

NCT05128825·Phase 2·ZNTL
Recruiting

Primary endpoint: Objective Response Rate (ORR) defined by RECIST v1.1 [Part 2]

InterventionalRandomizedopen310 targetStarted 2022-02Completion 2027-0650 sites · Australia, United StatesK-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

A Phase 1/2 Dose-Escalation and Dose-Expansion Study of ZN-c3 in Combination With Niraparib and ZN-c3 Monotherapy in Subjects With Platinum-Resistant Ovarian Cancer

NCT05198804·Phase 1/Phase 2·ZNTL
Completed

Primary endpoint: To investigate the safety and tolerability of ZN-c3 in combination with niraparib, including identification of the MTD and RP2D

Interventionalopen117 enrolledStarted 2022-01Completion 2026-0122 sites · France, United StatesK-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

A Phase 1/2 Dose Escalation and Dose Expansion Study of ZN-c3 in Combination With Gemcitabine in Adult and Pediatric Subjects With Relapsed or Refractory Osteosarcoma

NCT04833582·Phase 1·ZNTL
Completed

Primary endpoint: Incidence of dose-limiting toxicities (DLT) in DLT evaluable subjects and the incidence and severity of adverse events.

Interventionalopen31 enrolledStarted 2021-08Completion 2024-0317 sites · France, United StatesK-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

A Phase 2 Open-Label, Multicenter Study to Evaluate Efficacy and Safety of ZN-c3 in Adult Women With Recurrent or Persistent Uterine Serous Carcinoma

NCT04814108·Phase 2·ZNTL
Completed

Primary endpoint: Frequency and severity of TEAEs

Interventionalopen92 enrolledStarted 2021-07Completion 2025-1050 sites · Australia, Canada, United StatesK-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

A Phase 1b Study of ZN-c3 in Combination With Chemotherapy or Bevacizumab in Subjects With Ovarian, Peritoneal, or Fallopian Tube Cancer

NCT04516447·Phase 1·ZNTL
Recruiting

Primary endpoint: Part 1: To investigate the safety and tolerability of azenosertib in combination with PLD, carboplatin, paclitaxel, or gemcitabine

Interventionalopen172 targetStarted 2020-10Completion 2028-0624 sites · Australia, Bosnia and Herzegovina, Bulgaria, Georgia…K-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

A Phase 1 Study of ZN-c3 as a Single Agent in Subjects With Solid Tumors

NCT04158336·Phase 1·ZNTL
Completed

Primary endpoint: Dose Escalation

InterventionalRandomizedopen274 enrolledStarted 2019-11Completion 2025-058 sites · United StatesK-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

A Window of Opportunity Strategy for Targeted Pathway Inhibition in Patients With Pancreatic Ductal Adenocarcinoma

NCT04005690·Early Phase 1
Recruiting

Primary endpoint: Proportion of all pharmacodynamic feasibility-evaluable participants within a study arm that have a measurable change in post-treatment tumor biology from baseline

Interventionalopen90 targetStarted 2019-08Completion 2028-021 site · United StatesOHSU Knight Cancer Institute

Frequently asked questions

Who is developing azenosertib?

azenosertib is being developed by Zentalis Pharmaceuticals, Inc..

How many clinical trials involve azenosertib?

BioSniper tracks 9 clinical trials involving azenosertib.